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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50220706'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50220706((R)-N-((S)-1-(4-benzyl-4-((1-methyl-1H-tetrazol-5-...)
Affinity DataIC50:  52nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50220706((R)-N-((S)-1-(4-benzyl-4-((1-methyl-1H-tetrazol-5-...)
Affinity DataEC50:  111nMAssay Description:Antagonist activity at human MC4R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed