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Found 3 Enz. Inhib. hit(s) with Target = 'Vascular endothelial growth factor receptor 3' and Ligand = 'BDBM50363397'
TargetVascular endothelial growth factor receptor 3(Mus musculus (mouse))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of mouse VEGFR-3 (818 to 1363 residues)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Shanghai AB PharmaTech Ltd.

US Patent
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)
Affinity DataIC50: >10nMAssay Description:In this experiment, the inhibitory effects of small molecule inhibitors on 17 kinases were examined by using fluorescent microfluidic mobility shift ...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Shanghai AB PharmaTech Ltd.

US Patent
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)
Affinity DataIC50:  46nMAssay Description:Inhibition of VEGFR3 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank