Report error Found 6 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50307117'
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.74nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1a receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.74nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14.1nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at V1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Activity at human vasopressin V1a receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair