Report error Found 2030 with Last Name = 'zhu' and Initial = 'by'
Affinity DataKi: 0.000350nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.000570nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.000870nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.00150nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.00170nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.00200nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.00940nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0120nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Tested for binding affinity against human Coagulation factor Xa (trypsin-like serine protease)More data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Inhibitory activity of the compound against Coagulation factor Xa (serine protease) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.0350nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0830nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0830nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of human JAK2 (828-1132) expressed in baculovirus-infected Sf9 cells using EQEDEPEGDYFEWLE as substrate after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibitory activity of the compound against factor Xa,activity expressed as Ki nMMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human JAK1 (837-1142) expressed in baculovirus-infected Sf9 cells using EQEDEPEGDYFEWLE as substrate after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Apparent binding affinity to PI3Kalpha using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human GST-fused JAK3 catalytic domain expressed in baculovirus-infected Sf9 cells using polyglutamic acid-tyrosine as substrate after 3...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Coagulation factor XMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of recombinant PI3Kalpha assessed as inhibition of PIP3 formation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair