Report error Found 3763 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk1'
Affinity DataKi: 0.180nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.299nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 1.36nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 1.75nM ΔG°: -49.5kJ/molepH: 7.4 T: 22°CAssay Description:The inhibitors reported in this study bind to CHK1 according to a general mechanism illustrated in Scheme 1 where E, S, and I stand for enzyme, subst...More data for this Ligand-Target Pair
Affinity DataKi: 2.95nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 3.93nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 4.38nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 4.57nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 5.14nM ΔG°: -46.5kJ/molepH: 8.0 T: 20°CAssay Description:Surface plasmon resonance (SPR) biosensor binding studies were conducted using a Biacore 3000 instrument (GE Healtchare).More data for this Ligand-Target Pair
Affinity DataKi: 5.17nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 5.22nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
Affinity DataKi: 5.26nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair