TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Hebrew University Of Jerusalem
Curated by ChEMBL
Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at TRPV1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 69nMAssay Description:Agonist activity at rat CB1 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 minsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Hebrew University Of Jerusalem
Curated by ChEMBL
Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Hebrew University Of Jerusalem
Curated by ChEMBL
Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Hebrew University Of Jerusalem
Curated by ChEMBL
Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Activation of human VR1 expressed in HEK293 cells assessed as stimulation of Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+4nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+4nMAssay Description:Cannabinoid receptor 1 dependent activity of compound was evaluated by using [35S]GTP-gamma-S-binding studiesMore data for this Ligand-Target Pair