TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 535nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 537nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 8.04E+3nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 8.13E+3nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair