Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of ic50 for monomerid = 50268725
TargetP2X purinoceptor 2(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  588nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  2.22E+3nMAssay Description:Antagonist activity against human P2Y4 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  2.37E+3nMAssay Description:Antagonist activity at human P2Y4 receptor expressed in astrocytoma cells assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  3.16E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  4.63E+3nMAssay Description:Antagonist activity against human P2Y2 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  4.63E+3nMAssay Description:Antagonist activity at human P2Y2 receptor expressed in astrocytoma cells assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  5.30E+3nMAssay Description:Antagonist activity at rat P2Y6 receptor expressed in astrocytoma cells assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  5.30E+3nMAssay Description:Antagonist activity against human P2Y6 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed