TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of FLAG-tagged DDR1 in human HEK293 cells assessed as reduction in collagen-1-induced DDR1 phosphorylation incubated for 18 hrs by ELISAMore data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Vanderbilt University
Curated by ChEMBL
Vanderbilt University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of kinase tracer 178 binding to recombinant human GST-tagged DDR1 expressed in baculovirus expression system incubated for 60 mins by TR-F...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:The enzymatic activities DDR2 were tested in LanthaScreen binding assays. The protocol is available from Life Technologies.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of kinase tracer 178 binding to recombinant human GST-tagged DDR2 (427-855 residues) expressed in baculovirus expression system incubated ...More data for this Ligand-Target Pair
Affinity DataIC50: 753nMAssay Description:The enzymatic activities DDR2 were tested in LanthaScreen binding assays. The protocol is available from Life Technologies.More data for this Ligand-Target Pair