Affinity DataIC50: 27nMAssay Description:Antagonist activity at OX2 receptor assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Antagonist activity at OX1 receptor assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair