Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ki for monomerid = 104689
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human OX2 receptor in cell membrane by in vitro radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at human OX2R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
Merch Sharp & Dohme

US Patent
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  0.240nMAssay Description:Radioligand binding assay described in Bergman et. al. Bioorg. Med. Chem. Lett. 2008, 18, 1425-1430.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))TBA
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human OX1R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))TBA
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  1nMAssay Description:Binding affinity to human OX1 receptor in cell membrane by in vitro radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Rattus norvegicus (Rat))
Merch Sharp & Dohme

US Patent
LigandPNGBDBM104689(US8569311, A-9)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay described in Bergman et. al. Bioorg. Med. Chem. Lett. 2008, 18, 1425-1430.More data for this Ligand-Target Pair
In DepthDetails US Patent