Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ki for monomerid = 50001515
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of 1 nM [3H]- N6-(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Pharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  5.90E+4nMAssay Description:Binding affinity against Adenosine A2 receptor in rat striatal membranes using [3H]5'-(N-ethylcarboxamido)-adenosine (NECA) as the ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  1.33E+5nMAssay Description:Affinity against adenosine A2 receptor in brain membranes by displacement of [3H]CPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  1.56E+5nMAssay Description:Inhibition of c-AMP phosphodiesterase activity in guinea pig tracheal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  2.40E+5nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed