Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50001515'
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Pharmazeutische Chemie

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  5.90E+4nMAssay Description:Binding affinity against Adenosine A2 receptor in rat striatal membranes using [3H]5'-(N-ethylcarboxamido)-adenosine (NECA) as the ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  1.33E+5nMAssay Description:Affinity against adenosine A2 receptor in brain membranes by displacement of [3H]CPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50001515(1-Methylxanthine (1-Mx) | 3-Methyl-3,7-dihydro-pur...)
Affinity DataKi:  2.40E+5nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed