Affinity DataKi: 0.210nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Alpha-1-adrenergic receptor binding affinity of the compound, value taken from literatureMore data for this Ligand-Target Pair
Affinity DataKi: 0.269nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic alpha1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.269nMAssay Description:Binding affinity to adrenergic alpha1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.288nMAssay Description:Displacement of [125I]BE2254 from human cloned adrenergic alpha 1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.363nMAssay Description:Binding affinity to adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.363nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic Alpha-1D receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.363nMAssay Description:Displacement of [125I]BE2254 from human cloned adrenergic alpha 1D receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]BE2254 from human cloned adrenergic alpha 1B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.82nMAssay Description:Binding affinity to adrenergic Alpha-1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.82nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic Alpha-1B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A in CRL:CD(SD)BR-COBS rat brain hippocampus after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor measured by displacing [3H]-8-OH-DPAT from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor in human periipheral mononuclear leukocyte membranes using [125I]-pindololMore data for this Ligand-Target Pair