Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ki for monomerid = 50014732
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  10nMAssay Description:Compound was evaluated In vitro for inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  88nMAssay Description:Binding affinity against human Cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  110nMAssay Description:Binding affinity against human ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi: >6.00E+5nMAssay Description:Binding affinity against human Cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  1.00E+6nMAssay Description:Binding affinity against human ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed