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Found 3 Enz. Inhib. hit(s) with Target = 'Neutrophil elastase' and Ligand = 'BDBM50014732'
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against human Elastase for more active diasteriomerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  10nMAssay Description:Compound was evaluated In vitro for inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylami...)
Affinity DataKi:  110nMAssay Description:Binding affinity against human ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed