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Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM166905'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM166905(US9073870, 201)
Affinity DataIC50:  149nMpH: 6.0 T: 2°CAssay Description:In vitro inhibition of 11beta -HSD1 by test compounds was determined with HTRF (Homogeneous Time-Resolved Fluorescence) technology (cisbio internatio...More data for this Ligand-Target Pair
In DepthDetails US Patent