Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM50244290'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50244290(2-(2-bromo-6-ethoxy-4-((3-mercapto-5-methyl-4H-pyr...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of human recombinant 11beta-HSD1 expressed in HEK293 cell lysate assessed as conversion of radiolabeled estrone to estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed