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Found 2 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM50334705'
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Korea University

Curated by ChEMBL
LigandPNGBDBM50334705(3-Benzenesulfonyl-thiazolidine-2-carboxylic acid(5...)
Affinity DataIC50:  6nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 3 hrs by HTRF cortisol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50334705(3-Benzenesulfonyl-thiazolidine-2-carboxylic acid(5...)
Affinity DataIC50:  67nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO cells after 3 hrs by HTRF cortisol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed