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Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM57506'
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM57506((5R,9R,10R,13S,14S,17S)-4,4,10,13,14-pentamethyl-1...)
Affinity DataIC50:  880nMAssay Description:Inhibition of mouse microsomal 11beta-HSD1 overexpressed in HEK293 cells using [3H]-cortisone as substrate assessed as formation of [3H]-cortisol usi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed