Found 1 Enz. Inhib. hit(s) with Target = '17-beta-hydroxysteroid dehydrogenase type 1' and Ligand = 'BDBM50353136'
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq - Research Center And Laval University
Curated by ChEMBL
Chuq - Research Center And Laval University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 17beta-HSD1 in human T47D cells expressing estrogen receptor assessed as conversion of [14C]-E1 to [14C]-E2 after 24 hrsMore data for this Ligand-Target Pair