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Found 3 Enz. Inhib. hit(s) with Target = '17-beta-hydroxysteroid dehydrogenase type 2' and Ligand = 'BDBM25851'
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25851(3-[5-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  745nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25851(3-[5-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  745nMAssay Description:Inhibition of human placental 17betaHSD2 by radiodetection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25851(3-[5-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  745nMAssay Description:Inhibition of human placental 17beta-HSD2 microsomal fraction using tritiated estradiol as substrate assessed as formation of estrone by HPLC analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed