Found 1 Enz. Inhib. hit(s) with Target = '3-phosphoinositide-dependent protein kinase 1' and Ligand = 'BDBM104016'
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt
Universit£Tsklinikum Frankfurt
Affinity DataIC50: 3.80E+4nMpH: 7.4 T: 2°CAssay Description:A 20ul mix containing 50mM Tris pH 7.5, 0.05mg/ml BSA, 0.1% β-mercaptoethanol, 10mM MgCl2, 100μM [γ-P32]ATP (5-50cpm/pmol), 0.003% Bri...More data for this Ligand-Target Pair