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Found 2 Enz. Inhib. hit(s) with Target = '3-phosphoinositide-dependent protein kinase 1' and Ligand = 'BDBM50125790'
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Bioinformatics Institute (Bii)

Curated by ChEMBL
LigandPNGBDBM50125790(CHEMBL3623846)
Affinity DataKd:  3.94E+4nMAssay Description:Displacement of PIFtide from human PDK1 PIF pocket after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Bioinformatics Institute (Bii)

Curated by ChEMBL
LigandPNGBDBM50125790(CHEMBL3623846)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of human PDK1 catalytic activity using PIFtide as substrate after 1 hr by phosphor imager analysis in presence of [gamma-32P]-ATP relative...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed