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Found 4 Enz. Inhib. hit(s) with Target = '5'-AMP-activated protein kinase catalytic subunit alpha-1' and Ligand = 'BDBM50434272'
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50434272(CHEMBL1242297)
Affinity DataEC50:  8.00E+3nMAssay Description:Activation of human recombinant AMPK alpha1 subunitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50434272(CHEMBL1242297)
Affinity DataEC50:  9.00E+3nMAssay Description:Activation of human AMPK alpha1 (1 to 394) expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50434272(CHEMBL1242297)
Affinity DataEC50:  9.60E+3nMAssay Description:Activation of recombinant AMPK alpha1 (1 to 394) (unknown origin) after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50434272(CHEMBL1242297)
Affinity DataEC50:  8.00E+3nMAssay Description:Activation of human recombinant AMPK alpha1 (1 to 394 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL using SAMS peptide after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed