Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50005132'
Affinity DataKi: 13nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to 5-HT1A (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences
Curated by ChEMBL
Polish Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:In vitro ability to displace [3H]-8-hydroxy-2-(di-n-propylamino) tetralin binding from 5-hydroxytryptamine 1A receptor site in rat brain hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy of Sciences
Curated by ChEMBL
Polish Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Evaluated for binding affinity towards 5-hydroxytryptamine 1A receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataEC50: 288nMAssay Description:Activity against 5HT1A receptor by Gi-[35S]GTPgammaS binding assayMore data for this Ligand-Target Pair