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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50054366'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054366(2-[4-(4-Phenyl-piperazin-1-yl)-butyl]-tetrahydro-i...)
Affinity DataKi:  78.5nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054366(2-[4-(4-Phenyl-piperazin-1-yl)-butyl]-tetrahydro-i...)
Affinity DataKi:  79nMAssay Description:Tested in vitro for binding affinity by measuring its ability to inhibit [3H]8-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat cerebral cor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054366(2-[4-(4-Phenyl-piperazin-1-yl)-butyl]-tetrahydro-i...)
Affinity DataKi:  79nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor in rat cerebral cortex membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails Article