Found 15 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1B' and Ligand = 'BDBM50007406'
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity of the compound in radioreceptor binding assay by using [3H]-5-HT radioligand against 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Intrinsic affinity of the compound towards serotonin receptor from rat frontal cortex by displacement of [3H]-5-HTMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 298nMAssay Description:Intrinsic affinity of the compound towards serotonin receptor from rat frontal cortex by displacement of [3H]-spiperone.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1B receptor of rat cortex using [3H]-5-HTMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Concentration of the compound necessary to achieve half maximal inhibition of [125I]- Iodocyanopindolol binding to 5-hydroxytryptamine 1B receptor at...More data for this Ligand-Target Pair