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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1B' and Ligand = 'BDBM50456732'
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456732(CHEMBL4207355)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]5-CT from human 5-HT1B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456732(CHEMBL4207355)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456732(CHEMBL4207355)
Affinity DataEC50:  180nMAssay Description:Partial agonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed