Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2' and Ligand = 'BDBM235962'
Target5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2(Human)
Confluence Life Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 235962BDBM235962(US9365546, 285)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:Kinase reactions is carried out in a 384-well plate (Matrical, MP101-1-PP) in 20 mM HEPES pH 7.5, 10 mM MgCl2, 0.0005% Tween-20, 0.01% BSA, 1 mM DTT,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2(Human)
Confluence Life Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 235962BDBM235962(US9365546, 285)
Affinity DataIC50: 26nMpH: 7.5 T: 2°CAssay Description:Kinase reactions is carried out in a 384-well plate (Matrical, MP101-1-PP) in 20 mM HEPES pH 7.5, 10 mM MgCl2, 0.0005% Tween-20, 0.01% BSA, 1 mM DTT,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2(Human)
Confluence Life Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 235962BDBM235962(US9365546, 285)
Affinity DataIC50: 121nMpH: 7.5 T: 2°CAssay Description:Kinase reactions is carried out in a 384-well plate (Matrical, MP101-1-PP) in 20 mM HEPES pH 7.5, 10 mM MgCl2, 0.0005% Tween-20, 0.01% BSA, 1 mM DTT,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A/MAP kinase-activated protein kinase 2(Human)
Confluence Life Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 235962BDBM235962(US9365546, 285)
Affinity DataIC50: 210nMpH: 7.5 T: 2°CAssay Description:Kinase reactions is carried out in a 384-well plate (Matrical, MP101-1-PP) in 20 mM HEPES pH 7.5, 10 mM MgCl2, 0.0005% Tween-20, 0.01% BSA, 1 mM DTT,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent