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Found 8 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM35920'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of radioligand are dispensed into the wells of 96-well plates. Then, duplicate aliquots of the test and reference compound dilutions are add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2A receptor expressed NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor expressed NIH3T3 cells using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor sites by using [3H]-Ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM35920(9,10-dihydroanthracene(DHA), 1a | 9-(Aminomethyl)-...)
Affinity DataKi:  20nMAssay Description:Binding affinity of the compound was performed using [3H]-ketanserin as the radioligand and stably transfected NIH3T3 cells expressing the 5-hydroxyt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed