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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50145626'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50145626(CHEMBL3765122)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50145626(CHEMBL3765122)
Affinity DataIC50:  1.17E+3nMAssay Description:Antagonist activity at 5HT2A receptor in Sprague-Dawley rat ileum assessed as inhibition of 5-HT-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed