Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50145626'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£
Curated by ChEMBL
Dipartimento Di Farmacia Universit£
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£
Curated by ChEMBL
Dipartimento Di Farmacia Universit£
Curated by ChEMBL
Affinity DataIC50: 1.17E+3nMAssay Description:Antagonist activity at 5HT2A receptor in Sprague-Dawley rat ileum assessed as inhibition of 5-HT-induced contractionMore data for this Ligand-Target Pair