Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50604193'
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity to 5-HT2B receptor (unknown origin) assessed as displacement of radioligand at 10 uM by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) transfected in HEK293 cells assessed as beta-arrestin translocation by Tango assayMore data for this Ligand-Target Pair