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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50036718'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50036718(4-Phenyl-1,2,3,6-tetrahydro-pyridine | 4-phenyl-1,...)
Affinity DataKi:  7.18E+3nMAssay Description:Displacement of [3H]-mesulergine from 5HT2C receptor expressed in CHO cell membranes after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50036718(4-Phenyl-1,2,3,6-tetrahydro-pyridine | 4-phenyl-1,...)
Affinity DataEC50:  2.45E+3nMAssay Description:Agonist activity at 5HT2C receptor expressed in CHO cells by fluorescence based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed