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Found 5 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50076245'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50076245(CHEMBL1628670 | US10544152, Cpd # 1 | WAY-163909)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]DOI from human 5-HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50076245(CHEMBL1628670 | US10544152, Cpd # 1 | WAY-163909)
Affinity DataKi:  11nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50076245(CHEMBL1628670 | US10544152, Cpd # 1 | WAY-163909)
Affinity DataEC50:  18.2nMAssay Description:Cell Lines and Cell Culture.The PathHunter® U2OS HTR2C β-Arrestin cell line (5-HT2cR-U2OS; DiscoveRx) stably express the nonedited human 5-HT2CR...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50076245(CHEMBL1628670 | US10544152, Cpd # 1 | WAY-163909)
Affinity DataEC50:  8nMAssay Description:Agonist activity at 5HT2C receptor (unknown origin) relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50076245(CHEMBL1628670 | US10544152, Cpd # 1 | WAY-163909)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human 5-HT2C receptor assessed as stimulation of Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed