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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A/3B' and Ligand = 'BDBM50081989'
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50081989(5-(4-Methyl-piperazin-1-yl)-pyrazolo[1,5-c]quinazo...)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor from rat cortical homogenate using [3H]-zacopride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50081989(5-(4-Methyl-piperazin-1-yl)-pyrazolo[1,5-c]quinazo...)
Affinity DataEC50:  2.70nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed