Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50288284'
Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50288284BDBM50288284(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-iodo-2-...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for its binding affinity towards 5-hydroxytryptamine 3 receptor in whole rat brain using (S)-[125I]-zacopride as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50288284BDBM50288284(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-iodo-2-...)
Affinity DataKi:  1.40nMAssay Description:Compound was tested for its binding affinity towards 5-hydroxytryptamine 3 receptor in whole rat brain using [125I]DAIZAC as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50288284BDBM50288284(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-iodo-2-...)
Affinity DataKd:  2.60nMAssay Description:Compound was tested in vitro for its antagonistic activity against 5-hydroxytryptamine 3 receptor in rat CNS.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article