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Found 4 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50363325'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50363325(CHEMBL1945843)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]NAMH from human cloned 5HT3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50363325(CHEMBL1945843)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]NAMH from rat cloned 5HT3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50363325(CHEMBL1945843)
Affinity DataEC50:  1.10nMAssay Description:Antagonist activity at human recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50363325(CHEMBL1945843)
Affinity DataEC50:  1.60nMAssay Description:Antagonist activity at rat recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed