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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50398964'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Angelini Santa Palomba Research Center

Curated by ChEMBL
LigandPNGBDBM50398964(CHEMBL2179707)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H](1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate from human 5HT4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Angelini Santa Palomba Research Center

Curated by ChEMBL
LigandPNGBDBM50398964(CHEMBL2179707)
Affinity DataIC50:  9.80nMAssay Description:Antagonist activity at human 5HT4ER expressed in CHO cells assessed as reduction in cAMP levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed