Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50414730'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50414730(CHEMBL553404)
Affinity DataKi:  5.01nMAssay Description:Displacement of [H]GR-113808 from human 5HT4C receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50414730(CHEMBL553404)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at human 5HT4C receptor expressed in HEK293 cells assessed as acumulation of cAMP by flash plate adenylyl cyclase activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed