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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50515598'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Normandie Univ

Curated by ChEMBL
LigandPNGBDBM50515598(CHEMBL4526049)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to recombinant human brain 5HT4 receptor by radio ligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Normandie Univ

Curated by ChEMBL
LigandPNGBDBM50515598(CHEMBL4526049)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [3H]-GR 113808 from recombinant human brain 5HT4 receptor measured after 60 mins by radio ligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Normandie Univ

Curated by ChEMBL
LigandPNGBDBM50515598(CHEMBL4526049)
Affinity DataEC50:  2.80nMAssay Description:Partial agonist activity at human HA-tagged 5HT4 receptor expressed in COS7 cells assessed as induction of cAMP production measured after 10 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed