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Found 7 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50085970'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  20nMpH: 7.4Assay Description:The h5-HT6 radioligand binding assays were performed as previously described. In brief, h5-HT6 cDNA was transiently expressed in HEK-293 cells using...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  20nMAssay Description:Compound was evaluated for its binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  20nMAssay Description:Binding affinity against 5 Hydroxy tryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor transfected in HEK293 cells after 60 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  50nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Virginia Commonwealth University

LigandPNGBDBM50085970(CHEMBL7318 | [2-(5-Methoxy-2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  54nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptor expressed in HEK 293 human embryonic kidney cells, [3H]-lysergic acid diethylamide as radio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed