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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50304001'
Target5-hydroxytryptamine receptor 6(MOUSE)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50304001(CHEMBL584690 | [4-(4-Methylpiperazin-1-yl)-1H-benz...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50304001(CHEMBL584690 | [4-(4-Methylpiperazin-1-yl)-1H-benz...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50304001(CHEMBL584690 | [4-(4-Methylpiperazin-1-yl)-1H-benz...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed