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Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM86428'
Target5-hydroxytryptamine receptor 6(MOUSE)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM86428(SB-258585)
Affinity DataKi:  0.75nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86428(SB-258585)
Affinity DataKi:  1.82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(RAT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86428(SB-258585)
Affinity DataKi:  2.29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86428(SB-258585)
Affinity DataKi:  2.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(MOUSE)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM86428(SB-258585)
Affinity DataKi:  11.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86428(SB-258585)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at human 5-HT6 receptor expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP accumulation pretreated for 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed