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Found 9 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 7' and Ligand = 'BDBM50204672'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]D-lysergic acid diethylamide from 5HT7R (unknown origin) expressed in HEK293 cell membranes incubated for 1.5 hrs in absence of l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H] D-lysergic acid diethylamide from 5-HT7R (unknown origin) transfected in HEK293 cells incubated for 1.5 hrs by microbeta scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H] D-lysergic acid diethylamide from 5-HT7R (unknown origin) transfected in HEK293 cells incubated for 1.5 hrs by microbeta scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  148nMAssay Description:Agonist activity at 5-HT7R (unknown origin) transfected in HEK293 cells expressing tTA-dependent luciferase reporter and beta arrestin 2-TEV fusion g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  150nMAssay Description:Agonist activity at 5-HT7R (unknown origin) transfected in HEK293 cells expressing tTA-dependent luciferase reporter and beta arrestin 2-TEV fusion g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  457nMAssay Description:Agonist activity at human 5-HT7R transfected in HEK293 cells assessed as Gs-mediated cAMP accumulation incubated for 30 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human 5-HT7R transfected in HEK293 cells assessed as Gs-mediated cAMP accumulation incubated for 30 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  550nMAssay Description:Agonist activity at human 5-HT7R expressed in HEK293 cells assessed as induction of cAMP levels treated for 10 mins measured after 30 mins by D2-dye ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50204672(CHEMBL3961059)
Affinity DataEC50:  550nMAssay Description:Agonist activity at human 5-HT7R expressed in HEK293 cells assessed as induction of cAMP levels treated for 10 mins measured after 30 mins by D2-dye ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed