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Found 3 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase' and Ligand = 'BDBM50163799'
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50163799(5-Amino-3-(2-ethoxy-ethyl)-3-[4-(4-[1,3,4]oxadiazo...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against matrix metalloprotease 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50163799(5-Amino-3-(2-ethoxy-ethyl)-3-[4-(4-[1,3,4]oxadiazo...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant MMP2 using (Ac-PLG-[2-mercapto-4-85 methylpentanoyl]-LG-OC2H5) as substrate by microplate photometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50163799(5-Amino-3-(2-ethoxy-ethyl)-3-[4-(4-[1,3,4]oxadiazo...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant MMP2 using (Ac-PLG-[2-mercapto-4-85 methylpentanoyl]-LG-OC2H5) as substrate by microplate photometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed