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Found 3 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase' and Ligand = 'BDBM92443'
Target72 kDa type IV collagenase(Homo sapiens (Human))
Commissariat Á

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Commissariat Á

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi: >1.00E+3nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target72 kDa type IV collagenase(Homo sapiens (Human))
Commissariat Á

LigandPNGBDBM92443(MMP Inhibitor, 3 | Thiophene derivative, compound ...)
Affinity DataKi:  1.06E+3nM ΔG°:  -34.1kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using matrix metalloproteinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed