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Found 4 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 2' and Ligand = 'BDBM50391004'
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataKi:  2.58E+4nMAssay Description:TP_TRANSPORTER: inhibition of Temocaprilat uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataKi:  3.45E+4nMAssay Description:TP_TRANSPORTER: inhibition of 5-methyltetrahydrofolate uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataIC50:  1.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of Naf-GlcA uptake (Naf-GlcA: 0.1 uM) in bile canalicular membrane vesicles of Wistar ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataIC50:  1.93E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed