Found 4 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 2' and Ligand = 'BDBM58924'
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataKi: 5.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in canalicular membrane vesicles of rat liverMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in canalicular membrane vesicles of rat liverMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Deutsches Krebsforschungszentrum
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in Mrp2-expressing HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair