Found 3 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11' and Ligand = 'BDBM50190500'
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development
Curated by ChEMBL
Novo Nordisk Research And Development
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cells in presence of 2 mM ATPMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development
Curated by ChEMBL
Novo Nordisk Research And Development
Curated by ChEMBL
Affinity DataIC50: 3.60E+5nMAssay Description:Displacement of [3H]glibenclamide from human Kir6.2/SUR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development
Curated by ChEMBL
Novo Nordisk Research And Development
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Repolarization of HEK293 cells expressing Kir6.2/SUR1 KATP channelsMore data for this Ligand-Target Pair